About 20 results found for searched term "TA 01" (0.055 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M2154 | TAK-901 | Aurora Kinase |
| TAK901 | ||
| TAK-901 is a novel small-molecule inhibitor of Aurora A and Aurora B with IC50 of 21 nM and 15 nM. | ||
| M3274 | Pentagastrin | Cholecystokinin Receptor |
| Peptavlon; ICI-50123 | ||
| Pentagastrin (ICI-50123) is a synthetic polypeptide that has effects like gastrin when given parenterally. | ||
| M3729 | TAC-101 | CDK |
| Amsilarotene | ||
| TAC-101 is a retinobenzoic acid with potential antineoplastic activity. | ||
| M3973 | Tazarotene | RAR/RXR |
| Tazorac; Zorac; AGN 190168 | ||
| Tazarotene (AGN 190168) is a new member of the acetylenic class of RARβ/γ selective retinoids which is approved to treat a variety of skin diseases, exhibits an anti-proliferative effect in human basal cell carcinoma (BCC) by triggering caspase-dependent apoptosis. | ||
| M5291 | Sufugolix | LHRH/GnRH |
| TAK-013 | ||
| Sufugolix (TAK-013) is a highly potent and orally available luteinizing hormone-releasing hormone LHRH receptor antagonist with an IC50 of 0.1 nM. | ||
| M5928 | Riboflavin | Vitamin |
| Vitamin B2; E101 | ||
| Riboflavin is an easily absorbed micronutrient with a key role in maintaining health in humans and other animals. | ||
| M6070 | EDO-S101 | HDAC |
| Tinostamustine; EDO-S-101; EDO-S 101 | ||
| EDO-S101 is a pan HDAC inhibitor; inhibits HDAC1, HDAC2 and HDAC3 with IC50 values of 9, 9 and 25 nM, respectively. | ||
| M6140 | TA 01 | Casein Kinase |
| TA-01; TA01 | ||
| TA-01 potently inhibits CK1ε, CK1δ,and p38α (IC50values are 6.4, 6.8, and 6.7 nM respectively). | ||
| M7355 | TAS 301 | Others |
| TAS 301 is a inhibitor of smooth muscle cell migration and proliferation. | ||
| M9041 | PF-03084014 (Nirogacestat) | Gamma-secretase/Beta-secretase |
| Nirogacestat; PF-3084014 | ||
| PF-03084014 (Nirogacestat) is a potent and selective γ-secretase inhibitor with IC50 of 6.2 nM. | ||
| M9197 | Relugolix | LHRH/GnRH |
| Orgovyx; TAK-385; RVT-601 | ||
| Relugolix, also known as TAK-385, is an orally active gonadotropin-releasing hormone (GnRH) antagonist with an IC50 of 0.12 nM. | ||
| M11283 | Inolitazone dihydrochloride | PPAR |
| Efatutazone dihydrochloride; CS-7017 dihydrochloride; RS5444 dihydrochloride | ||
| Inolitazone dihydrochloride (Efatutazone dihydrochloride) is a PPARγ agonist with high affinity, activity dependent on PPARγ, inhibiting growth, IC50 is 0.8 nM. | ||
| M11549 | Palifosfamide | DNA Alkylator/Crosslinker |
| Isophosphoramide mustard; IPM; ZIO-201 | ||
| Palifosfamide(Isophosphoramide mustard; IPM; Zio-201) is a new DNA alkylation agent and active metabolite of isocyclophosphamide, which has anticancer activity. | ||
| M21064 | Bradanicline | Others |
| ATA-101; TC-5619 | ||
| Bradanicline (ATA-101; TC-5619) is a highly selective α7 nicotinic acetylcholine receptor (nAChR) agonist (EC50=17 nM for human α7 nAChR; Ki=1.4 nM). Bradanicline can be used to study cognitive impairment. | ||
| M24910 | Olinvacimab | VEGFR/PDGFR |
| TTAC-0001 | ||
| Olinvacimab (TTAC-0001) is a fully human anti-VEGFR2 monoclonal antibody. Olinvacimab inhibits VEGF binds to KDR with a Kd value of 0.23 nM. Olinvacimab has antiangiogenic activity. Olinvacimab can be used for the research of recurrent glioblastoma and breast cancer. | ||
| M25181 | Upanovimab | Others |
| SCTA01 | ||
| Upanovimab (SCTA01) is a monoclonal antibody. | ||
| M25429 | Rezafungin acetate | Anti-infection |
| Biafungin acetate; CD101 acetate; SP-3025 acetate | ||
| Rezafungin acetate is a novel echinocandin-based antifungal agent with potent antifungal activity against Candida, Aspergillus and Pneumocystis. | ||
| M28233 | Caficrestat | Aldose Reductase |
| Aldose reductase-IN-1; AT-001 | ||
| Caficrestat (Aldose reductase-IN-1) is a inhibitor of aldose reductase with IC50 of 28.9 pM. | ||
| M29393 | Inolitazone | PPAR |
| Efatutazone; CS-7017; RS5444 | ||
| Inolitazone a novel high-affinity PPARγ agonist that is dependent upon PPARγ for its biological activity with IC50 of 0.8 nM for growth inhibition. | ||
| M52383 | Tau Peptide (301-315) | Tau Protein |
| Tau Peptide (301-315) is a polypeptide that can be found by peptide screening. | ||
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